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Uptake inhibition assays were terminated by fast vacuum filtration by way of Whatman GF/B filters, and retained radioactivity was quantified by liquid scintillation counting. For release assays, nine nM [3H]MPP+ was used since the radiolabeled substrate for DAT and Internet, even though 5 nM [3H]serotonin was utilised as a substrate for SERT. A